Stereoselective synthesis of all stereoisomers of orthogonally protected cyclobutane-1,2-diamine and some chemoselective transformations

Research output: Contribution to journalArticleResearchpeer-review

16 Citations (Scopus)

Abstract

The four stereoisomers of protected cyclobutane-1,2-diamine have been prepared in an enantio- and diastereocontrolled manner through stereodivergent synthetic routes starting from a half-ester as a common chiral precursor. Orthogonal protection allows the chemoselective manipulation of both amino groups as shown in this work. © 2012 American Chemical Society.
Original languageEnglish
Pages (from-to)2431-2433
JournalOrganic Letters
Volume14
Issue number10
DOIs
Publication statusPublished - 18 May 2012

Fingerprint Dive into the research topics of 'Stereoselective synthesis of all stereoisomers of orthogonally protected cyclobutane-1,2-diamine and some chemoselective transformations'. Together they form a unique fingerprint.

  • Cite this