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Indolylarylsulfones carrying a heterocyclic tail as very potent and broad spectrum HIV-1 non-nucleoside reverse transcriptase inhibitors

Valeria Famiglini, Giuseppe La Regina, Antonio Coluccia, Sveva Pelliccia, Andrea Brancale, Giovanni Maga, Emmanuele Crespan, Roger Badia, Eva Riveira-Muñoz, José A. Esté, Rosella Ferretti, Roberto Cirilli, Claudio Zamperini, Maurizio Botta, Dominique Schols, Vittorio Limongelli, Bruno Agostino, Ettore Novellino, Romano Silvestri

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Pharmacology, Toxicology and Pharmaceutical Science

Biochemistry, Genetics and Molecular Biology